11. Novel drug discovery strategies for atherosclerosis that target necrosis and necroptosis. (3rd June 2018) Authors: Coornaert, Isabelle; Hofmans, Sam; Devisscher, Lars; Augustyns, Koen; Van Der Veken, Pieter; De Meyer, Guido R.Y.; Martinet, Wim Journal: Expert opinion on drug discovery Issue: Volume 13:Number 6(2018:Jun.) Page Start: 477 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
12. Novel selective glucocorticoid receptor agonists (SEGRAs) with a covalent warhead for long-lasting inhibition. Issue 20 (15th October 2016) Authors: Ryabtsova, Oksana; Joossens, Jurgen; Van Der Veken, Pieter; Vanden Berghe, Wim; Augustyns, Koen; De Winter, Hans Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 20(2016) Page Start: 5032 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
13. Preclinical evaluation of [111In]MICA‐401, an activity‐based probe for SPECT imaging of in vivo uPA activity. (24th August 2016) Authors: Vangestel, Christel; Thomae, David; Van Soom, Jeroen; Ides, Johan; wyffels, Leonie; Pauwels, Patrick; Stroobants, Sigrid; Van der Veken, Pieter; Magdolen, Viktor; Joossens, Jurgen; Augustyns, Koen; Staelens, Steven Journal: Contrast media & molecular imaging Issue: Volume 11:Number 6(2016:Nov./Dec.) Page Start: 448 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
14. Probing for improved selectivity with dipeptide-derived inhibitors of dipeptidyl peptidases 8 and 9: the impact of P1-variation. Issue 3 (26th November 2015) Authors: Heirbaut, Leen; van Goethem, Sebastiaan; Jansen, Koen; de Winter, Hans; Lamoen, Nicole; Joossens, Jurgen; Cheng, Jonathan; Chen, Xin; Lambeir, Anne-Marie; de Meester, Ingrid; Augustyns, Koen; van der Veken, Pieter Journal: MedChemComm Issue: Volume 7:Issue 3(2016:Mar.) Page Start: 433 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
15. Repositioning the Substrate Activity Screening (SAS) Approach as a Fragment‐Based Method for Identification of Weak Binders. Issue 15 (25th August 2014) Authors: Gladysz, Rafaela; Cleenewerck, Matthias; Joossens, Jurgen; Lambeir, Anne‐Marie; Augustyns, Koen; Van der Veken, Pieter Journal: Chembiochem Issue: Volume 15:Issue 15(2014) Page Start: 2238 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
16. Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity. (April 2019) Authors: Botros, Sanaa S.; William, Samia; Sabra, Abdel-Nasser A.; El-Lakkany, Naglaa M.; Seif el-Din, Sayed H.; García-Rubia, Alfonso; Sebastián-Pérez, Victor; Blaazer, Antoni R.; de Heuvel, Erik; Sijm, Maarten; Zheng, Yang; Salado, Irene G.; Munday, Jane C.; Maes, Louis; de Esch, Iwan J.P.; Sterk, Geert... Journal: International journal for parasitology Issue: Volume 9(2019) Page Start: 35 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
17. Selected strategies to fight pathogenic bacteria. (31st December 2023) Authors: Plotniece, Aiva; Sobolev, Arkadij; Supuran, Claudiu T.; Carta, Fabrizio; Björkling, Fredrik; Franzyk, Henrik; Yli-Kauhaluoma, Jari; Augustyns, Koen; Cos, Paul; De Vooght, Linda; Govaerts, Matthias; Aizawa, Juliana; Tammela, Päivi; Žalubovskis, Raivis Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 38:Number 1(2023) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
18. Selected strategies to fight pathogenic bacteria. (31st December 2023) Authors: Plotniece, Aiva; Sobolev, Arkadij; Supuran, Claudiu T.; Carta, Fabrizio; Björkling, Fredrik; Franzyk, Henrik; Yli-Kauhaluoma, Jari; Augustyns, Koen; Cos, Paul; De Vooght, Linda; Govaerts, Matthias; Aizawa, Juliana; Tammela, Päivi; Žalubovskis, Raivis Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 38:Number 1(2023) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
19. Structures of purine nucleosidase from Trypanosoma brucei bound to isozyme‐specific trypanocidals and a novel metalorganic inhibitor. (30th July 2013) Authors: Giannese, Francesca; Berg, Maya; Van der Veken, Pieter; Castagna, Valeria; Tornaghi, Paola; Augustyns, Koen; Degano, Massimo Journal: Acta crystallographica Issue: Volume 69:Part 8(2013:Aug.) Page Start: 1553 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
20. Substrate Activity Screening (SAS) and Related Approaches in Medicinal Chemistry. (4th February 2016) Authors: Gladysz, Rafaela; Lambeir, Anne‐Marie; Joossens, Jurgen; Augustyns, Koen; Van der Veken, Pieter Journal: ChemMedChem Issue: Volume 11:Number 5(2016) Page Start: 467 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗