1. Identification and optimisation of 4, 5-dihydrobenzo[1, 2-d:3, 4-d]bisthiazole and 4, 5-dihydrothiazolo[4, 5-h]quinazoline series of selective phosphatidylinositol-3 kinase alpha inhibitors. Issue 17 (1st September 2015) Authors: Fairhurst, Robin A.; Gerspacher, Marc; Imbach-Weese, Patricia; Mah, Robert; Caravatti, Giorgio; Furet, Pascal; Fritsch, Christine; Schnell, Christian; Blanz, Joachim; Blasco, Francesca; Desrayaud, Sandrine; Guthy, Daniel A.; Knapp, Mark; Arz, Dorothee; Wirth, Jasmin; Roehn-Carnemolla, Esther; Luu... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 17(2015) Page Start: 3575 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Identification and optimisation of a 4′, 5-bisthiazole series of selective phosphatidylinositol-3 kinase alpha inhibitors. Issue 17 (1st September 2015) Authors: Fairhurst, Robin A.; Imbach-Weese, Patricia; Gerspacher, Marc; Caravatti, Giorgio; Furet, Pascal; Zoller, Thomas; Fritsch, Christine; Haasen, Dorothea; Trappe, Joerg; Guthy, Daniel A.; Arz, Dorothee; Wirth, Jasmin Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 17(2015) Page Start: 3569 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗