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Author/Creator Andrys, Rudolf

1. 1, 2, 4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy. (1st January 2020)

Authors:
Kaproń, Barbara; Czarnomysy, Robert; Wysokiński, Mariusz; Andrys, Rudolf; Musilek, Kamil; Angeli, Andrea; Supuran, Claudiu T.; Plech, Tomasz
Journal:
Journal of enzyme inhibition and medicinal chemistry
Issue:
Volume 35:Number 1(2020)
Page Start:
993
Record Type:
Journal Article
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2. Charged pyridinium oximes with thiocarboxamide moiety are equally or less effective reactivators of organophosphate-inhibited cholinesterases compared to analogous carboxamides. (31st December 2022)

Authors:
Kohoutova, Zuzana; Malinak, David; Andrys, Rudolf; Svobodova, Jana; Psotka, Miroslav; Schmidt, Monika; Prchal, Lukas; Musilek, Kamil
Journal:
Journal of enzyme inhibition and medicinal chemistry
Issue:
Volume 37:Number 1(2022)
Page Start:
760
Record Type:
Journal Article
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3. Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition. (1st January 2021)

Authors:
Oleksak, Patrik; Psotka, Miroslav; Vancurova, Marketa; Sapega, Olena; Bieblova, Jana; Reinis, Milan; Rysanek, David; Mikyskova, Romana; Chalupova, Katarina; Malinak, David; Svobodova, Jana; Andrys, Rudolf; Rehulkova, Helena; Skopek, Vojtech; Ngoc Lam, Pham; Bartek, Jiri; Hodny, Zdenek; Musilek, K...
Journal:
Journal of enzyme inhibition and medicinal chemistry
Issue:
Volume 36:Number 1(2021)
Page Start:
410
Record Type:
Journal Article
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4. Encapsulation of oxime K027 into cucurbit[7]uril: In vivo evaluation of safety, absorption, brain distribution and reactivation effectiveness. (1st March 2020)

Authors:
Zdarova Karasova, Jana; Hepnarova, Vendula; Andrys, Rudolf; Lisa, Miroslav; Jost, Petr; Muckova, Lubica; Pejchal, Jaroslav; Herman, David; Jun, Daniel; Kassa, Jiri; Kuca, Kamil
Journal:
Toxicology letters
Issue:
Volume 320(2020)
Page Start:
64
Record Type:
Journal Article
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5. Privileged multi-target directed propargyl-tacrines combining cholinesterase and monoamine oxidase inhibition activities. (31st December 2022)

Authors:
Chrienova, Zofia; Nepovimova, Eugenie; Andrys, Rudolf; Dolezal, Rafael; Janockova, Jana; Muckova, Lubica; Fabova, Lenka; Soukup, Ondrej; Oleksak, Patrik; Valis, Martin; Korabecny, Jan; Marco-Contelles, José; Kuca, Kamil
Journal:
Journal of enzyme inhibition and medicinal chemistry
Issue:
Volume 37:Number 1(2022)
Page Start:
2605
Record Type:
Journal Article
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6. Pyridinium-2-carbaldoximes with quinolinium carboxamide moiety are simultaneous reactivators of acetylcholinesterase and butyrylcholinesterase inhibited by nerve agent surrogates. (1st January 2021)

Authors:
Lee, Hyun Myung; Andrys, Rudolf; Jonczyk, Jakub; Kim, Kyuneun; Vishakantegowda, Avinash G.; Malinak, David; Skarka, Adam; Schmidt, Monika; Vaskova, Michaela; Latka, Kamil; Bajda, Marek; Jung, Young-Sik; Malawska, Barbara; Musilek, Kamil
Journal:
Journal of enzyme inhibition and medicinal chemistry
Issue:
Volume 36:Number 1(2021)
Page Start:
437
Record Type:
Journal Article
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7. Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators. (1st January 2020)

Authors:
Malinak, David; Dolezal, Rafael; Hepnarova, Vendula; Hozova, Miroslava; Andrys, Rudolf; Bzonek, Petr; Racakova, Veronika; Korabecny, Jan; Gorecki, Lukas; Mezeiova, Eva; Psotka, Miroslav; Jun, Daniel; Kuca, Kamil; Musilek, Kamil
Journal:
Journal of enzyme inhibition and medicinal chemistry
Issue:
Volume 35:Number 1(2020)
Page Start:
478
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗