Search

Author/Creator Altman, Michael D.

1. Corrigendum to "Design of selective PI3Kδ inhibitors using an iterative scaffold-hopping workflow" [Bioorg. Med. Chem. Lett. 29 (2019) 2575–2580]. Issue 16 (15th August 2020)

Authors:
Fradera, Xavier; Methot, Joey L.; Achab, Abdelghani; Christopher, Matthew; Altman, Michael D.; Zhou, Hua; McGowan, Meredeth A.; Kattar, Sam D.; Wilson, Kevin; Garcia, Yudith; Augustin, Martin A.; Lesburg, Charles A.; Shah, Sanjiv; Goldenblatt, Peter; Katz, Jason D.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 16(2020)
Page Start:
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

3. Design of selective PI3Kδ inhibitors using an iterative scaffold-hopping workflow. Issue 18 (15th September 2019)

Authors:
Fradera, Xavier; Methot, Joey L.; Achab, Abdelghani; Christopher, Matthew; Altman, Michael D.; Zhou, Hua; McGowan, Meredeth A.; Kattar, Sam D.; Wilson, Kevin; Garcia, Yudith; Augustin, Martin A.; Lesburg, Charles A.; Shah, Sanjiv; Goldenblatt, Peter; Katz, Jason D.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 18(2019)
Page Start:
2575
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

4. Development of a High-Throughput Gene Expression Screen for Modulators of RAS-MAPK Signaling in a Mutant RAS Cellular Context. (October 2016)

Authors:
Severyn, Bryan; Nguyen, Thi; Altman, Michael D.; Li, Lixia; Nagashima, Kumiko; Naumov, George N.; Sathyanarayanan, Sriram; Cook, Erica; Morris, Erick; Ferrer, Marc; Arthur, Bill; Benita, Yair; Watters, Jim; Loboda, Andrey; Hermes, Jeff; Gilliland, D. Gary; Cleary, Michelle A.; Carroll, Pamela M.;...
Journal:
SLAS discovery
Issue:
Volume 21:Number 9(2016)
Page Start:
989
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

5. Discovery of a new series of PI3K-δ inhibitors from Virtual Screening. (15th June 2021)

Authors:
Fradera, Xavier; Deng, Qiaolin; Achab, Abdelganhi; Garcia, Yudith; Kattar, Solomon D.; McGowan, Meredeth A.; Methot, Joey L.; Wilson, Kevin; Zhou, Hua; Shaffer, Lynsey; Goldenblatt, Peter; Tong, Vincent; Augustin, Martin A; Altman, Michael D.; Lesburg, Charles A.; Shah, Sanjiv; Katz, Jason D.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 42(2021)
Page Start:
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

6. Identification of N-(1H-pyrazol-4-yl)carboxamide inhibitors of interleukin-1 receptor associated kinase 4: Bicyclic core modifications. Issue 22 (15th November 2015)

Authors:
Lim, Jongwon; Altman, Michael D.; Baker, James; Brubaker, Jason D.; Chen, Hongmin; Chen, Yiping; Kleinschek, Melanie A.; Li, Chaomin; Liu, Duan; Maclean, John K.F.; Mulrooney, Erin F.; Presland, Jeremy; Rakhilina, Larissa; Smith, Graham F.; Yang, Ruojing
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 22(2015)
Page Start:
5384
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

7. Identification of quinazoline based inhibitors of IRAK4 for the treatment of inflammation. Issue 12 (15th June 2017)

Authors:
Smith, Graham F.; Altman, Michael D.; Andresen, Brian; Baker, James; Brubaker, Jason D.; Chen, Hongmin; Chen, Yiping; Childers, Matthew; Donofrio, Anthony; Ferguson, Heidi; Fischer, Christian; Fischmann, Thierry O.; Gibeau, Craig; Hicks, Alexander; Jin, Sue; Kattar, Sam; Kleinschek, Melanie A.; L...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 12(2017)
Page Start:
2721
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

8. MARK inhibitors: Declaring a No-Go decision on a chemical series based on extensive DMPK experimentation. Issue 1 (1st January 2017)

Authors:
Haidle, Andrew M.; Childers, Kaleen K.; Zabierek, Anna A.; Katz, Jason D.; Jewell, James P.; Hou, Yongquan; Altman, Michael D.; Szewczak, Alexander; Chen, Dapeng; Harsch, Andreas; Hayashi, Mansuo; Warren, Lee; Hutton, Michael; Nuthall, Hugh; Stanton, Matt G.; Davies, Ian W.; Munoz, Ben; Northrup,...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 1(2017)
Page Start:
109
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

9. Optimization of microtubule affinity regulating kinase (MARK) inhibitors with improved physical properties. Issue 17 (1st September 2016)

Authors:
Sloman, David L.; Noucti, Njamkou; Altman, Michael D.; Chen, Dapeng; Mislak, Andrea C.; Szewczak, Alexander; Hayashi, Mansuo; Warren, Lee; Dellovade, Tammy; Wu, Zhenhua; Marcus, Jacob; Walker, Deborah; Su, Hua-Poo; Edavettal, Suzanne C.; Munshi, Sanjeev; Hutton, Michael; Nuthall, Hugh; Stanton, M...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 17(2016)
Page Start:
4362
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

10. Structure guided design of a series of selective pyrrolopyrimidinone MARK inhibitors. Issue 1 (1st January 2017)

Authors:
Katz, Jason D.; Haidle, Andrew; Childers, Kaleen K.; Zabierek, Anna A.; Jewell, James P.; Hou, Yongquan; Altman, Michael D.; Szewczak, Alexander; Chen, Dapeng; Harsch, Andreas; Hayashi, Mansuo; Warren, Lee; Hutton, Michael; Nuthall, Hugh; Su, Hua-Poo; Munshi, Sanjeev; Stanton, Matt G.; Davies, Ia...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 1(2017)
Page Start:
114
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗