1. Discovery of 1, 8-naphthyridin-2-one derivative as a potent and selective sphingomyelin synthase 2 inhibitor. Issue 7 (1st April 2020) Authors: Yukawa, Takafumi; Nakahata, Takashi; Okamoto, Rei; Ishichi, Yuji; Miyamoto, Yasufumi; Nishimura, Satoshi; Oikawa, Tatsuo; Kubo, Kazuki; Adachi, Ryutaro; Satomi, Yoshinori; Nakakariya, Masanori; Amano, Nobuyuki; Kamaura, Masahiro; Matsunaga, Nobuyuki Journal: Bioorganic & medicinal chemistry Issue: Volume 28:Issue 7(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of Human Intestinal MGAT Inhibitors Using High-Throughput Mass Spectrometry. (April 2017) Authors: Adachi, Ryutaro; Ishii, Tsuyoshi; Matsumoto, Shinichi; Satou, Takuya; Sakamoto, Junichi; Kawamoto, Tomohiro Journal: SLAS discovery Issue: Volume 22:Number 4(2017) Page Start: 360 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of novel serine palmitoyltransferase inhibitors as cancer therapeutic agents. Issue 9 (15th May 2018) Authors: Kojima, Takuto; Asano, Yasutomi; Kurasawa, Osamu; Hirata, Yasuhiro; Iwamura, Naoki; Wong, Tzu-Tshin; Saito, Bunnai; Tanaka, Yuta; Arai, Ryosuke; Yonemori, Kazuko; Miyamoto, Yasufumi; Sagiya, Yoji; Yaguchi, Masahiro; Shibata, Sachio; Mizutani, Akio; Sano, Osamu; Adachi, Ryutaro; Satomi, Yoshinori;... Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 9(2018) Page Start: 2452 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Inhibition of MGAT2 modulates fat‐induced gut peptide release and fat intake in normal mice and ameliorates obesity and diabetes in ob/ob mice fed on a high‐fat diet. Issue 3 (5th February 2020) Authors: Mochida, Taisuke; Take, Kazumi; Maki, Toshiyuki; Nakakariya, Masanori; Adachi, Ryutaro; Sato, Kenjiro; Kitazaki, Tomoyuki; Takekawa, Shiro Journal: FEBS open bio Issue: Volume 10:Issue 3(2020) Page Start: 316 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities. Issue 15 (1st August 2015) Authors: Sato, Kenjiro; Takahagi, Hiroki; Kubo, Osamu; Hidaka, Kousuke; Yoshikawa, Takeshi; Kamaura, Masahiro; Nakakariya, Masanori; Amano, Nobuyuki; Adachi, Ryutaro; Maki, Toshiyuki; Take, Kazumi; Takekawa, Shiro; Kitazaki, Tomoyuki; Maekawa, Tsuyoshi Journal: Bioorganic & medicinal chemistry Issue: Volume 23:Issue 15(2015) Page Start: 4544 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Using a biologically annotated library to analyze the anticancer mechanism of serine palmitoyl transferase (SPT) inhibitors. Issue 4 (13th February 2017) Authors: Sano, Osamu; Kazetani, Ken‐ichi; Adachi, Ryutaro; Kurasawa, Osamu; Kawamoto, Tomohiro; Iwata, Hidehisa Journal: FEBS open bio Issue: Volume 7:Issue 4(2017) Page Start: 495 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗